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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1197 | Sincalide | SQ19844,CCK-8,Cholecystokinin octapeptide | Others |
Sincalide (CCK-8) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. It is the 8-amino acid C-terminal fragment of cholecystokinin. | |||
TP1198 | Sincalide ammonium | SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium | cholecystokinin |
Sincalide ammonium (CCK-8 ammonium) is a potent analog of the amino acid peptide hormone cholecystokinin (CCK), an active fragment that retains much of the biological activity of CCK.Sincalide ammonium promotes bile secr... | |||
T9343 | N-Cbz-DL-tryptophan | cholecystokinin | |
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8. | |||
TP1931L1 | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate | [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) | cholecystokinin |
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ... | |||
T25108 | ARL 15849XX | ARL15849XX,FPL15849,FPL-15849,FPL 15849,ARL-15849XX | |
ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent. | |||
T34669 | Snf 8906 | Snf-8906,Snf8906 | |
Snf 8906 is a CCK-8 analog. | |||
T25437 | Fpl 14294 | Fpl-14294,Fpl14294 | |
Fpl 14294 is a novel CCK-8 agonist with effective intranasal anorectic activity in the rat. | |||
T16906 | Sograzepide | YM-220,Netazepide,YF 476 | Others |
Sograzepide is an effective and highly selective Gastrin/CCK-B antagonist (IC50: 0.1 nM), has an inhibitory effect on Gastrin/CCK-A activity (IC50: 502 nM). Sograzepide replaces the specific binding of [125I]CCK-8 to the... | |||
T15105 | Dexloxiglumide | Others | |
Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors. | |||
T60700 | Butabindide | ||
Butabindide (UCL-1397) is a potent, selective inhibitor of tripeptidvl peptidase II (TPP II) with Ki values of 10 μM and 7 nM for TPP I and TPP II, respectively. Butabindide inhibits TPP II in order to protect CCK-8 agai... | |||
T36629 | Givinostat | ||
Givinostat (ITF-2357) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. Givinostat (ITF2357) suppresses total LPS-induced IL-1β production robustly compared with the reduction by ITF30... |